Pyrimidine derivatives, process for preparing the same and agric

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

Patent

Rate now

  [ 0.00 ] – not rated yet Voters 0   Comments 0

Details

514272, 544321, 544330, 544332, A61K 31505, C07D23942, C07D23946, A01N 4354

Patent

active

049924389

ABSTRACT:
Disclosed are pyrimidine derivatives represented by general formula (I) ##STR1## wherein X represents a hydrogen atom, a halogen atom, an alkyl group, an alkoxy group, a haloalkyl group or a cyano group; Y.sup.1 represents an alkyl group, a cyanoalkyl group, an alkoxy group, an alkenyl group substituted with a hydroxy group and a halogen atom, an alkynyl group which may be substituted with a hydroxy group, a methylamino group, an alkoxyalkyloxy group, an alkylthioalkyl group or a group of the formula --CH.sub.2 OR.sup.1 where R.sup.1 represents a hydrogen atom, an alkyl group, an alkenyl group or an alkynyl group; Y.sup.2 represents a halogen atom, an alkyl group or a haloalkyl group; R represents a hydrogen atom, an alkyl group, a nitroso group, an alkoxyalkyl group, an alkoxyalkyloxyalkyl group, an alkenyl group, an alkynyl group, a formyl group or an alkylthioalkyl group, with the proviso that (a) when Y.sup.1 represents an alkynyl grop or when Y.sup.1 represents an alkoxy group and Y.sup.2 represents a halogen atom or an alkyl group, X and R are not a hydrogen atom simultaneously, (b) when Y.sup.1 and Y.sup.2 each represents an alkyl group, R is not a hydrogen atom, or (c) when Y.sup.1 represents an alkyl group and Y.sup.2 represents a halogen atom, X and R are not a hydrogen atom simultaneously or X is not a halogen atom nor an alkyl group. Also, agricultural or horticultural compositions containing the pyrimidine derivatives as active ingredient are disclosed, which show high controlling activities for cucumber gray mold (Botrytis cinerea), cucumber downey mildew (Pseudoperonospora cubensis), Alternaria sooty spot of Chineese mustard (Alternaria brassicicola), rice blast (Pyricularia oryzae), etc.

REFERENCES:
patent: 3974276 (1976-08-01), Barlow et al.
patent: 3980781 (1976-09-01), Snell et al.
patent: 4082535 (1978-04-01), Hoegerle et al.
patent: 4092150 (1978-05-01), Treves
patent: 4248618 (1981-02-01), Serban et al.
patent: 4248619 (1981-02-01), Serban et al.
patent: 4814338 (1989-03-01), Ito et al.
Franke et al., CA, 96-157395n, (1982), "Fungicidal Compositions Containing Pyrimidines".
Serban et al., CA 94-65716y, (1981).
Ito et al., CA 104-168491a, (1986).
Evers et al., CA 104-148917r, (1986).

LandOfFree

Say what you really think

Search LandOfFree.com for the USA inventors and patents. Rate them and share your experience with other people.

Rating

Pyrimidine derivatives, process for preparing the same and agric does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Pyrimidine derivatives, process for preparing the same and agric, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Pyrimidine derivatives, process for preparing the same and agric will most certainly appreciate the feedback.

Rate now

     

Profile ID: LFUS-PAI-O-20760

  Search
All data on this website is collected from public sources. Our data reflects the most accurate information available at the time of publication.