Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Patent
1995-11-08
1998-04-21
Ivy, C. Warren
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
514211, 514212, 514218, 5142278, 5142372, 514307, 514311, 514314, 514315, 514318, 514319, 514326, 514343, 514345, 514374, 514422, 514423, 540480, 540481, 540483, 540544, 540553, 540575, 540597, 540602, 540596, 540603, 540607, 540610, 546145, 546146, 546153, 546187, 546194, 546206, 546207, 546208, 546209, 546210, 546212, 546214, 546245, 5462791, 548146, 548212, 5483147, 548517, 548537, 548538, 548572, A61K 31445, A61K 3140, C07D40112, C07D20709, C07D21128
Patent
active
057417997
ABSTRACT:
Heterocyclic thrombin inhibitors are provided which have the structure ##STR1## wherein n, R, R.sup.1, R.sup.2, R.sup.3, G, G.sub.x, R.sup.6', Ra, Xa, R.sup.6, Rb, R.sub.3, p, Q, A and R.sup.4 are as defined herein.
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Das Jagabandhu
Hall Steven E.
Han Wen-Ching
Kimball Spencer D.
Lau Wan Fang
Bristol--Myers Squibb Company
Huang Evelyn
Ivy C. Warren
Rodney Burton
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