Process for preparing pharmaceutically active compounds and inte

Details Process for preparing pharmaceutically active compounds and inte Process for preparing pharmaceutically active compounds and inte

1997-11-10

2000-11-28

Dentz, Bernard

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

546115, 546223, C07D21122, C07D21158, C07D49804

Patent

active

061537551

ABSTRACT:
##STR1## A process is disclosed for the preparation of (1) by reduction of (2) directly using catalytic transfer hydrogenation to suppress formation of (4) or by conventional reduction via (4). Compound (1) is a key intermediate for inter alia paroxetine.

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