Organic compounds -- part of the class 532-570 series – Organic compounds – Heterocyclic carbon compounds containing a hetero ring...
Patent
1989-10-03
1991-05-14
Waddell, Frederick E.
Organic compounds -- part of the class 532-570 series
Organic compounds
Heterocyclic carbon compounds containing a hetero ring...
546282, C07D40104
Patent
active
050157418
ABSTRACT:
This invention provides a novel class of nicotine analogs which as therapeutic agents exhibit tranquilizing effects in mammals.
Illustrative of invention nicotine analogs are 1-(3-dimethylaminopropyl)-2-(3-pyridyl)pyrrolidine: ##STR1## and (R,S)-6-(N,N-dimethyl-3-aminopropyl)nicotine: ##STR2## The nicotine analogs can exist in the form of acid addition salts.
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Osdene Thomas S.
Secor Henry V.
Seeman Jeffrey I.
DePaoli George A.
Kilby Scalzo Catherine S.
Philip Morris Incorporated
Schardt James E.
Waddell Frederick E.
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