Tricyclic steroid receptor modulator compounds and methods

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

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514242, 514243, 514246, 514247, 514248, 514249, 514250, 514255, 514256, 514259, 514292, 514411, 544179, 544180, 544183, 544233, 544234, 544235, 544238, 544245, 544246, 544249, 544284, 544338, 544342, 544343, 544344, 544353, 546 81, 546 84, 546 89, 546 92, 548432, A61K 3144, A61K 3147, A61K 3140, C07D47152, C07D47104

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056961308

ABSTRACT:
Non-steroidal compounds which are high affinity, high selectivity modulators for steroid receptors are disclosed. Also disclosed are pharmaceutical compositions incorporating such compounds, methods for employing the disclosed compounds and compositions for treating patients requiring steroid receptor agonist or antagonist therapy, intermediates useful in the preparation of the compounds and processes for the preparation of the steroid receptor modulator compounds.

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