Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...
Patent
1999-08-17
2000-11-21
Shah, Mukund J.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Heterocyclic carbon compounds containing a hetero ring...
5142335, 51425214, 5142522, 51425301, 51425309, 51425401, 51425411, 514226, 514320, 514337, 514364, 514397, 514422, 514456, 540575, 544151, 544277, 544295, 544376, 546196, 5462831, 548131, 5483114, 548525, 549399, 549404, C07D21542, C07D31168, A61K 31352
Patent
active
061503568
ABSTRACT:
Indanes, benzopyrans and analogues thereof are potassium channel inhibitors and blockers of IKur and have the structure ##STR1## where A, B, D, Q, X.sup.1, R, R.sup.1, X.sup.2 and R.sup.2 are as defined herein. These compounds are useful as antiarrhythmic agents. In addition, a method is provided for preventing cardiac arrhythmia employing the above compounds.
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Atwal Karnail S.
Finlay Heather J.
Gross Michael F.
Lloyd John
Spear Kerry L.
Bristol--Myers Squibb Company
Rao Deepak R.
Rodney Burton
Shah Mukund J.
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