Hindered esters of rapamycin

Details Hindered esters of rapamycin Hindered esters of rapamycin

1993-11-22

1995-01-31

Bond, Robert T.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

540456, A61K 31445, C07D47104

Patent

active

053859081

ABSTRACT:
A compound of the structure ##STR1## wherein R and R.sup.1 are each, independently, ##STR2## or hydrogen; R.sup.2 and R.sup.3 are each, independently, alkyl, arylalkyl, or R.sup.2 and R.sup.3 may be taken together to form a cycloalkyl ring;

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