Carboxyalkyl tricyclic derivatives useful as inhibitors of enkep

Details Carboxyalkyl tricyclic derivatives useful as inhibitors of enkep Carboxyalkyl tricyclic derivatives useful as inhibitors of enkep

1993-11-02

1995-10-03

Shah, Mukund J.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Heterocyclic carbon compounds containing a hetero ring...

540521, 540522, A61K 3155, C07D49804

Patent

active

054552427

ABSTRACT:
The present invention relates to compounds of the formula ##STR1## wherein B.sub.1 and B.sub.2 are each independently hydrogen; hydroxy; --OR.sub.2 wherein R.sub.2 is a C.sub.1 -C.sub.4 alkyl or an Ar--Y group wherein Ar is aryl and Y is a hydrogen or C.sub.1 -C.sub.4 alkyl; or, where B.sub.1 and B.sub.2 are attached to adjacent carbon atoms, B.sub.1 and B.sub.2 can be taken together with said adjacent carbons to form a benzene ring or methylenedioxy;

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