Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Patent
1992-05-29
1993-09-21
Dentz, Bernard
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
546133, A61K 31435, C07D45302
Patent
active
052469425
ABSTRACT:
This invention is directed to certain dibenzofurancarboxamides and their use as 5HT.sub.3 antagonists having unique CNS, anti-emetic and gastric prokinctic activity void of any significant D.sub.2 receptor binding properties. This invention also describes novel processes necessary for their preparation.
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Airey John E.
Campbell Henry F.
Klein Scott I.
Kuhla Donald E.
Powers Matthew R.
Dentz Bernard
Rhone-Poulenc Rorer Pharmaceuticals Inc.
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