Water soluble prodrugs of secondary and tertiary amine containin

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Phosphorus containing other than solely as part of an...

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514 85, 514100, 514114, 540542, 544337, 549220, 558166, 558203, 558131, A61K 31675, A61K 31665, A61K 3166, C07F 96561, C07F 96509

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active

059858567

ABSTRACT:
The present invention is drawn to water soluble derivatives aliphatic acid aromatic secondary and tertiary amine containing drugs. The present invention is further drawn to methods of making water soluble derivatives of aliphatic and aromatic secondary and tertiary amine containing drugs.

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