Water soluble adenosine kinase inhibitors

Details Water soluble adenosine kinase inhibitors Water soluble adenosine kinase inhibitors

1995-06-07

1998-03-10

Wilson, James O.

Organic compounds -- part of the class 532-570 series

Organic compounds

Carbohydrates or derivatives

536 272, 536 276, 536 2761, 536 2762, 536 2763, 536 277, C07H 1916

Patent

active

057263027

ABSTRACT:
This invention relates to adenosine kinase inhibitors and to nucleoside analogs, specifically to water soluble, aryl substituted 4-amino analogs having activity as adenosine kinase inhibitors. The invention also relates to the preparation and use of these adenosine kinase inhibitors in the treatment of cardiovascular, and cerebrovascular diseases, inflammation and other diseases which can be regulated by increasing the local concentration of adenosine.

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