Use of saccharin derivatives as proteolytic enzyme inhibitors

Details Use of saccharin derivatives as proteolytic enzyme inhibitors Use of saccharin derivatives as proteolytic enzyme inhibitors

1993-05-24

1994-12-06

Brust, Joseph Paul

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Silicon containing doai

514 80, 5142242, 5142342, 514242, 514274, 514253, 514373, 514363, 514361, 514339, 514314, 514 32, 514364, 514369, A61K 31425, A61K 31535

Patent

active

053710746

ABSTRACT:
Novel 2-substituted saccharins which inhibit the enzymatic activity of proteolytic enzymes, are useful in the treatment of degenerative diseases and have the formula 0010
wherein:

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