Use of phthalazine derivatives

Details Use of phthalazine derivatives Use of phthalazine derivatives

2005-06-07

2005-06-07

Richter, Johann (Department: 1626)

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Heterocyclic carbon compounds containing a hetero ring...

C544S237000

Reexamination Certificate

active

06903098

ABSTRACT:
The present invention relates to the use of phthalazine derivatives as inhibitors of the enzyme poly(ADP-ribose) polymerase or PARP (EC 2.4.2.30), to the use as inhibitors of PARP-homologous enzymes and, in particular, these phthalazine derivatives also show a selective inhibition of PARP-homologous enzymes.

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