Use of isoxazole and crotonamide derivatives for the treatment o

Details Use of isoxazole and crotonamide derivatives for the treatment o Use of isoxazole and crotonamide derivatives for the treatment o

1996-10-16

1999-03-23

Goldberg, Jerome D.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Ester doai

514522, A61K 31275

Patent

active

058860339

ABSTRACT:
The use of isoxazole and crotonamide derivatives for the treatment of carcinomatous disorders
The compound of the formula I or II ##STR1## is suitable for the production of a pharmaceutical for the treatment of carcinomatous disorders, where R.sup.1 is (C.sub.3 -C.sub.5)-cycloalkyl, (C.sub.2 -C.sub.6)-alkenyl or (C.sub.2 -C.sub.6)-alkynyl, R.sup.2 is CF.sub.3, OCF.sub.3, SCF.sub.3, OH, NO.sub.2, halogen, benzyl, phenyl, CN or O-phenyl, R.sup.3 is (C.sub.1 -C.sub.4)-alkyl, halogen or a hydrogen atom and X is a --CH group or a nitrogen atom.

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