Use of 7-alkylidene cephalosporins to inhibit elastase activity

Details Use of 7-alkylidene cephalosporins to inhibit elastase activity Use of 7-alkylidene cephalosporins to inhibit elastase activity

1996-12-06

1998-06-02

Shah, Mukund J.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Heterocyclic carbon compounds containing a hetero ring...

540215, 540223, 540228, 540230, 514202, 514209, C07D50120, A61K 31545

Patent

active

057600279

ABSTRACT:
The present invention relates to the use of 7-alkylidene derivatives of cephalosporin esters, such as sulfides, sulfoxides, and sulfones, as inhibitors of human leukocyte elastase. These materials are therefore useful as anti-inflammatory and anti-degenerative agents.

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