Unsymmetrical cyanine dimer compounds and their application

Chemistry: analytical and immunological testing – Fluorescent dyes

Reexamination Certificate

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C536S026600, C435S006120, C422S067000

Reexamination Certificate

active

07888136

ABSTRACT:
Embodiments of the present invention provide methods and nucleic acid reporter molecules for the detection of nucleic acid in a sample. The nucleic acid reporter molecule comprises two unsymmetrical cyanine monomer moieties, which may be the same or different, that are covalently attached by a linker comprising at least one aromatic, heteroaromatic, cyclic or heterocyclic moiety comprising 3-20 non-hydrogen atoms selected from the group consisting of O, N, S, P and C. The linker may be rigid, relatively flexible or some degree thereof. The unsymmetrical cyanine monomer moieties comprise a substituted or unsubstituted benzazolium moiety and a substituted or unsubstituted pyridinium or quinolinium moiety that is connected by a methine bridge that is monomethine, trimethine or pentamethine. The linkers form the cyanine dimer compounds by attaching to the pyridinium or quinolinium moiety of the monomer moieties. The present nucleic acid reporter molecules find utility in forming a nucleic acid-reporter molecule complex and detecting the nucleic acid. In particular, present nucleic acid reporter molecules with a rigid linker and monomer moieties with a monomethine bridge find utility in detecting RNA in the presence of DNA.

REFERENCES:
patent: 4711955 (1987-12-01), Ward et al.
patent: 4883867 (1989-11-01), Lee et al.
patent: 4957870 (1990-09-01), Lee et al.
patent: 5047519 (1991-09-01), Hobbs et al.
patent: 5314805 (1994-05-01), Haugland et al.
patent: 5352803 (1994-10-01), Mattingly
patent: 5362628 (1994-11-01), Haugland et al.
patent: 5410030 (1995-04-01), Yue et al.
patent: 5436134 (1995-07-01), Haugland et al.
patent: 5534416 (1996-07-01), Millard et al.
patent: 5545535 (1996-08-01), Roth et al.
patent: 5573904 (1996-11-01), Mattingly
patent: 5582977 (1996-12-01), Yue et al.
patent: 5658751 (1997-08-01), Yue et al.
patent: 5714327 (1998-02-01), Houthoff et al.
patent: 5863753 (1999-01-01), Haugland et al.
patent: 5929227 (1999-07-01), Glazer et al.
patent: 5963753 (1999-10-01), Ohtani et al.
patent: 6428667 (2002-08-01), Glazer et al.
patent: 6579718 (2003-06-01), Yue et al.
patent: 6664047 (2003-12-01), Haugland et al.
patent: 63-132688 (1988-06-01), None
patent: 02084383 (1990-03-01), None
patent: 2000-319260 (2000-11-01), None
patent: WO-93/06482 (1993-04-01), None
patent: WO-00/66664 (2000-11-01), None
patent: WO-2005/012579 (2005-02-01), None
Stratagene CATALOG 1988, p. 39.
Bunkenborg et al. Bioconjugate Chem. 2000, 11, 861-867.
U.S. Appl. No. 10/911,423, “Office Action mailed Sep. 17, 2007”.
U.S. Appl. No. 10/911,423, “Office Action mailed Dec. 21, 2007”.
U.S. Appl. No. 10/911,423, “Response to Sep. 17, 2007 Office Action”, Filed Oct. 17, 2007.
U.S. Appl. No. 10/911,423, “Response to Rest. Req. Filed Jul. 9, 2007”.
U.S. Appl. No. 10/911,423, “Restriction Req. mailed Jun. 8, 2007”.
Brinkley, Michael, “A Brief Survey of Methods for Preparing Protein Conjugates with Dyes, Haptens, and Cross-Linking Reagents”,Bioconjugate Chem., vol. 3, No. 1 1992, 2-13.
Bunkenborg, Jakob et al., “Concerted intercalation and minor groove recognition of DNA by a homodimeric thiazole orange dye”,Bioconjugate Chemistryvol. 11, No. 6 Nov. 2000, 861-867.
Furniss, Brian S. et al., “Resolution of Racemates”,Vogel's Textbook of Practical Organic ChemistryFifth Ed, Longman Group UK Ltd., Essex 1989, 809-823.
Gaugain, Bernard, “DNA Bifunctional Intercalators 2. Fluorescence Properties and DNA Binding Interaction of an Ethidium Homodimer and an Acridine Ethidium Heterodimer”,Biochemistryvol. 17 No. 24 1978, 5078-5088.
Gaugain, Bernard et al., “DNA bifunctional intercalators. 1. Synthesis and conformational properties of an ethidium homodimer and of an acridine ethidium heterodimer”,Biochemistryvol. 17, No. 24 1978, 5071-5078.
Haugland, Richard P., “Molecular Probes Handbook of Fluorescent Probes and Research Products”,9th Edition, 2002(CD-Rom Format),Molecular Probes 2002.
Heller, A., “Electrical Wiring of Redox Enzymes”,Acc. Chem. Res. vol. 23, No. 5 1990, 128-134.
Hickman, David T. et al., “Kinetically selective binding of single stranded RNA over DNA by a pyrrolidine-amide oligonucleotide minic (POM)”,Nucleosides Nucleotides&Nucleic Acidsvol. 20, No. 4-7 2001, 1169-1172.
Markovits, J et al., “Dynamic Structure of DNA Complexes. Fluorometric Measurement of Hydrogen-Deuterium Exchange Kinetics of DNA-bound Ethidium Dimer and Acridine-Ethidium Dimer”,Biochemistryvol. 22, No. 13 1983, 3231-3237.
Markovits, Judith et al., “Effect of B-Z transition and nucleic add structure on the conformational dynamics of bound ethidium dimer measured by hydrogen deuterium exchange kinetics”,Nucl. Acids Res. 13 1985, 3773-3788.
Markovits, et al., “Ethidium Dimer: A New Reagent for the Fluorimetric Determination of Nucleic Acids”,Analytical Biochemistryvol. 94 1979 , 259-269.
Rye, Hays S. et al., “High-sensitivity two-color detection of double-stranded DNA with a confocal fluorescence gel scanner using ethidium homodimer and thiazole orange”,Nucleic Acids Resvol. 19 No. 2 1990, 327-333.
Sandler, Stanley R. et al., “Organic Functional Group Preparations”, vol. 3,New York: Academic Press1972, 5-7.
Singh, Tara et al., “Antimalarials. Distal Hydrazine derivatives of 7-chloroquinoline”,Journal of medicinal chemistryvol. 14, No. 6 1971, 532-5.
Staerk, Dan et al., “Bisintercalation of homodimeric thiazole orange dyes in DNA: Effect of modifying the linker”,Bioconjugate Chemistryvol. 8, No. 6 Nov. 1997, 869-877.
Stratagene Catalog 1988, “Stragagene Cloning Systems: Tools and Technology for Life Sciences”,Gene Characterization Kits1988, 39.
Timtcheva, I. et al., “Homodimeric monomethine cyanine dyes as fluorescent probes of biopolymers”,Journal of Photochemistry and Photobiology B Biologyvol. 58, No. 2-3 Nov. 2000, 130-135.
Yamana, Kazushige et al., “Bis-pyrene-labeled oligonucleotide: sequence specificity of excimer and monomer fluroescence changes upon hybridization with DNA”,Bioconjug Chemvol. 13, No. 6 2002, 1266-73.
Yamana, Kazushige et al., “Fluorescence Detection of Specific RNA Sequence Using 2′-Pyrene-Modified Oligoribonucleotides”,Angewandte Chemie International Edition in Englishvol. 40 No. 6 2001, 1104-1106.
WO 2005/012579, “International Report on Patentability”, Feb. 6, 2006.
WO 2005/012579, “PCT ISR”, Sep. 15, 2005.
WO 2005/012579, “Written Opinion of the International Searching Authority”, Jan. 31, 2006.

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