Tropane derivatives useful in therapy

Details Tropane derivatives useful in therapy Tropane derivatives useful in therapy

2007-04-04

2009-08-25

Andres, Janet L (Department: 1625)

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

Reexamination Certificate

active

07579471

ABSTRACT:
The present invention provides compounds of formula (I)wherein X, Y, R1, R2and R3are as defined hereinabove.The compounds of the present invention are modulators, especially antagonists, of the activity of chemokine CCR5 receptors. Modulators of the CCR5 receptor may be useful in the treatment of various inflammatory diseases and conditions, and in the treatment of infection by HIV and genetically related retroviruses.

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