Tritioacetylating reagents and processes for preparation thereof

Details Tritioacetylating reagents and processes for preparation thereof Tritioacetylating reagents and processes for preparation thereof

1998-10-23

2000-12-12

Wilson, James O.

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

548473, 548475, C07D20740

Patent

active

061601284

ABSTRACT:
Novel acetylating and tritioacetylating reagents suitable for preparation of nonlabelled and radiolabelled organic compounds. N-acetoxynaphthalimide, N-tritioacetoxyphthalimide, N-tritioacetoxysuccinimide, N-tritioacetoxynaphthalimide and processes of their preparation. The invention also concerns synthesis of nonlabelled acetylated and tritioacetylated organic compounds from precursors containing a free --NH.sub.2, --SH or --OH group.

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