Tricyclic compound having spiro union

Details Tricyclic compound having spiro union Tricyclic compound having spiro union

2006-10-17

2006-10-17

Tucker, Zachary C. (Department: 1624)

Organic compounds -- part of the class 532-570 series

Organic compounds

Unsubstituted hydrocarbyl chain between the ring and the -c-...

C540S455000, C540S466000, C540S490000, C540S502000, C544S006000, C544S070000, C544S071000, C544S230000, C544S231000

Reexamination Certificate

active

07122662

ABSTRACT:
This invention relates to tricyclic compounds having spiro union represented by the following formula (I) or its salt which is useful as a drug, and in particular, as an inhibitor for activated blood coagulation factor X, which can be administered orally and which exhibits strong anticoagulation action.The invention also relates to a pharmacophore which was derived from the compound and is useful in molecular designing of the FXa inhibitor.

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