Tricyclic benzodiazepines

Chemistry of carbon compounds – Miscellaneous organic carbon compounds – C-metal

Patent

Rate now

  [ 0.00 ] – not rated yet Voters 0   Comments 0

Details

260295R, 260295AM, 2602955R, 2602955A, C07D21324

Patent

active

040496678

ABSTRACT:
Tricyclic benzodiazepine derivatives ("A") bearing a hydroxylower alkyl substituent in the 1-position and a heterocyclic ring joined between positions 4 and 5 of the benzodiazepine moiety are described. The heterocyclic ring will contain the nitrogen atom appearing at position 4 of the benzodiazepine ring as well as the hetero atom, which may be either oxygen or nitrogen, attached to the carbon atom at the 5-position of the benzodiazepine ring. "A" bearing an oxygen atom in the new heterocyclic ring may be formed from the corresponding 4,5-unsaturated benzodiazepines by treatment with an epoxide compound in the presence of an acid catalyst. "A" bearing either a nitrogen or an oxygen atom in the new heterocyclic ring may be prepared by cyclization of the corresponding open compound. "A" are useful as sedative, muscle relaxant and anti-convulsant agents.

REFERENCES:
patent: 3835149 (1974-09-01), Renfroe

LandOfFree

Say what you really think

Search LandOfFree.com for the USA inventors and patents. Rate them and share your experience with other people.

Rating

Tricyclic benzodiazepines does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Tricyclic benzodiazepines, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Tricyclic benzodiazepines will most certainly appreciate the feedback.

Rate now

     

Profile ID: LFUS-PAI-O-670586

  Search
All data on this website is collected from public sources. Our data reflects the most accurate information available at the time of publication.