Tricyclic amines with central dopaminergic activity

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

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540101, 540110, A61K 31445, C07D22110

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active

046123164

ABSTRACT:
Compounds of the formula ##STR1## wherein C.sup.1 and N.sup.4 are in trans configuration to each other, wherein R and Y are defined herein below, as bases and pharmaceutically acceptable acid addition salts thereof, processes for their preparation and pharmaceutical preparations and methods of treatment employing such compounds. The compounds are useful for treatment of disorders in the central nervous system.

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Cannon, J., et al., Journal of Medicinal Chemistry, 1979, 22(4), pp. 341-347.
Cannon, J., et al., Journal of Medicinal Chemistry, 1976, 19(8), pp. 987-993.
Cannon, J., et al., Journal of Medicinal Chemistry, 1980, 23(1), pp. 1-5.
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