Tricycle steroid analogs

Details Tricycle steroid analogs Tricycle steroid analogs

1993-10-15

1994-09-06

Killos, Paul J.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

9,10-seco- cyclopentanohydrophenanthrene ring system doai

514169, 514562, A01N 4500, A01N 3700

Patent

active

053448260

ABSTRACT:
Novel tricyclic steriod analogs are disclosed which are 1H-benz[e]indene dodecahydro compounds that are useful for enhancing GABA-induced chloride currents at the GABA receptor/chloride ionophore complex and can be represented by the following structural formulas: ##STR1## wherein R.sub.1 =H or C.sub.1 -C.sub.4 alkyl or fluoroalkyl;

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