Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...
Reexamination Certificate
2005-01-11
2008-11-11
Rao, Deepak (Department: 1624)
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Heterocyclic carbon compounds containing a hetero ring...
C514S275000, C514S318000, C514S326000, C544S122000, C544S331000, C546S210000
Reexamination Certificate
active
07449462
ABSTRACT:
Compounds of formula (I),or pharmaceutically acceptable derivatives thereof, wherein:Het represents 2-pyridinyl or 2-pyrimidinyl;R1represents H, C1-3alkyl or a nitrogen-containing heterocyclic ring having 5 or 6 ring atoms;R2represents H, benzyl or C1-3alkyl; andR3represents H, methyl, methoxy or chloro;are useful for treating anxiety, cardiovascular disease (including angina, atherosclerosis, hypertension, heart failure, edema, hypernatremia), dysmenorrhoea (primary and secondary), endometriosis, emesis (motion sickness), intrauterine growth retardation, inflammation (including rheumatoid arthritis), mittlesmerchz, preclampsia, premature ejaculation, premature (preterm) labor and Raynaud's disease.
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Bryans Justin S.
Johnson Patrick S.
Ryckmans Thomas
Stobie Alan
Benson Gregg C.
Pfizer Inc.
Rao Deepak
Wichtowski John A.
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