Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Nitrogen containing other than solely as a nitrogen in an...
Patent
1997-01-16
1997-11-18
Raymond, Richard L.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Nitrogen containing other than solely as a nitrogen in an...
564353, A61K 31135, C07C21718
Patent
active
056888309
ABSTRACT:
This invention relates to a compound of the Formula I: ##STR1## as a racemic mixture and its individual enantiomers, in particular the (R)-enantiomer, and their pharmaceutically acceptable salts. These compounds are useful as sodium channel blockers, and are particularly useful for the alleviation of neuropathic pain.
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Berger Jacob
Flippin Lee Allen
Hunter John Cureton
Loughhead David Garrett
Weikert Robert James
Kaku Janet K.
Lewis Brian
Raymond Richard L.
Syntex (U.S.A.) Inc.
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