Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Radical -xh acid – or anhydride – acid halide or salt thereof...
Patent
1992-08-06
1995-08-15
Cintins, Marianne M.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Radical -xh acid, or anhydride, acid halide or salt thereof...
514130, 514143, 514510, 514569, 514572, 514602, 514709, 514732, A61K 31195
Patent
active
054419832
ABSTRACT:
A method for inhibiting cell infection by an enveloped virus, by administering to an infection site, a therapeutically effective amount of a calix(n)arene compound derivatized, at its ring positions meta to the bridge attachements to the ring, with polar substitutent having a terminal carboxylate, phosphate, or sulfonate groups, including esters and amides which are cleavable in vivo. The compound may be administered orally, or topically, e.g., for treatment of herpes virus.
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Chen Jen
Choy William
Hwang Kou M.
Liu Su-Ying
Qi You M.
Cintins Marianne M.
Dehlinger Peter J.
Genelabs Incorporated
Powers Vincent M.
Travers Russell
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