Transdermal delivery of (R)-3,3-diphenylpropylamin-monoestern

Details Transdermal delivery of (R)-3,3-diphenylpropylamin-monoestern Transdermal delivery of (R)-3,3-diphenylpropylamin-monoestern

2011-04-05

2011-04-05

Sullivan, Daniel M (Department: 1621)

Drug, bio-affecting and body treating compositions

Preparations characterized by special physical form

Matrices

C514S546000

Reexamination Certificate

active

07919117

ABSTRACT:
The invention relates to a device for transdermally administering a compound of formula (I), wherein A represents hydrogen or deuterium, R represents a group selected among C1-4alkyl, C3-10cycloalkyl, or phenyl, each of which can be substituted by C1-3alkoxy, fluoride, chlorine, bromine, iodine, nitro, amino, hydroxy, oxo, mercapto, or deuterium, the C atom marked by * (asterisk) being provided in the R configuration. The invention is characterized in that the compound of general formula (I) is provided in a polymer matrix and is released at a dose of 0.5 to 20 mg per day through human skin. The invention further relates to the use of said compounds of formula (I) for producing transdermal medicaments.

REFERENCES:
patent: 4675009 (1987-06-01), Hymes et al.
patent: 5271940 (1993-12-01), Cleary et al.
patent: 6425892 (2002-07-01), Southam et al.
patent: 6555129 (2003-04-01), Arth et al.
patent: 6638528 (2003-10-01), Kanios
patent: 6743441 (2004-06-01), Sanders et al.
patent: 6858650 (2005-02-01), Meese
patent: 6893655 (2005-05-01), Flanigan et al.
patent: 7230030 (2007-06-01), Meese et al.
patent: 7246486 (2007-07-01), Nakagawa et al.
patent: 2003/0157156 (2003-08-01), Hsu et al.
patent: 2004/0081683 (2004-04-01), Schacht et al.
patent: 0957073 (1999-11-01), None
patent: 2199525 (2003-02-01), None
patent: 93/23025 (1993-11-01), None
patent: 99/58478 (1999-11-01), None
patent: 01/35957 (2001-05-01), None
patent: 2004/089872 (2004-10-01), None

Affiliated with

Also associated with

Rating

Transdermal delivery of (R)-3,3-diphenylpropylamin-monoestern does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Transdermal delivery of (R)-3,3-diphenylpropylamin-monoestern, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Transdermal delivery of (R)-3,3-diphenylpropylamin-monoestern will most certainly appreciate the feedback.

Rate now

Comments { 0 }

Profile ID: LFUS-PAI-O-2643654