Transdermal antiandrogenic compositions and modulated process

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Ester doai

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514691, 514944, 514946, 514947, 514969, 424443, 424446, A01N 3710

Patent

active

054829704

ABSTRACT:
Novel compositions comprising an antiandrogenic compound of the formula ##STR1## wherein R is COR.sub.1 wherein R.sub.1 is loweralkyl and a vehicle comprising a metabolism modulator and a polar organic solvent, and a method of controlling the membrane permeation and metabolism of the compound thereof are disclosed.

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