Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Patent
2000-02-02
2000-11-07
Tsang, Cecilia
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
514 75, 514 91, 514142, 514359, 514381, 514382, 514425, 514428, 514538, 514541, 514542, 514603, 514608, 514617, 514620, 514646, 514784, 548253, 548254, 548255, 548542, 548547, 560429, 560430, 560433, 560442, 562 11, 562 14, 562 15, 562 16, 562 30, 562 44, 564163, A61K 31401, A61P 3100, A61P 3500, C07D20748
Patent
active
06143776&
ABSTRACT:
Tosylproline analogs of formula I, methods of making them, pharmaceutical compositions containing them, and methods for their use. The compounds are thymidylate synthase inhibitors; and are useful as anti-tumor agents and as anti-parasitics, anti-bacterials, anti-fungals, and anti-virals.
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Oswecki Jane C.
Sunesis Pharmaceuticals, Inc.
Tsang Cecilia
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