Thiophenyl and pyrrolyl azepines as serotonin 5-HT 2c...

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...

Reexamination Certificate

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C514S215000, C540S543000, C540S578000, C540S586000, C540S593000

Reexamination Certificate

active

07893051

ABSTRACT:
The present invention generally relates to a series of compounds, to pharmaceutical compositions containing the compounds, and to use of the compounds and compositions as therapeutic agents. More specifically, compounds of the present invention are thiophenyl and pyrrolyl azepine compounds. These compounds are serotonin receptor (5-HT2c) ligands and are useful for treating diseases, disorders, and conditions wherein modulation of the activity of serotonin receptors (5-HT2c) is desired (e.g. addiction, anxiety, depression, obesity, and others).

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Supplemental European Search Report for corresponding European Application No. EP 07 71 8077, Jul. 13, 2010.

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