Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...
Reexamination Certificate
2008-04-15
2008-04-15
Habte, Kahsay T. (Department: 1624)
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Heterocyclic carbon compounds containing a hetero ring...
C544S071000, C544S092000
Reexamination Certificate
active
07358246
ABSTRACT:
Thioamide compounds, and specifically, thioamide pyrrole compounds, and preparation thereof are provided. These thioamide compounds can be used as progesterone receptor modulators, in contraception, and in the treatment of progesterone-related maladies.
REFERENCES:
patent: 3536809 (1970-10-01), Applezweig
patent: 3598123 (1971-08-01), Zaffaroni
patent: 3845770 (1974-11-01), Theevwes et al.
patent: 3916899 (1975-11-01), Theevwes et al.
patent: 4008719 (1977-02-01), Theevwes et al.
patent: 4295987 (1981-10-01), Parks
patent: 4959217 (1990-09-01), Sanders et al.
patent: 5124455 (1992-06-01), Lombardo
patent: 5273752 (1993-12-01), Ayer et al.
patent: 5459151 (1995-10-01), Lombardo
patent: 5756127 (1998-05-01), Grizoni et al.
patent: 5817343 (1998-10-01), Burke
patent: 5854388 (1998-12-01), Harding et al.
patent: 6391907 (2002-05-01), Fensome et al.
patent: 6407101 (2002-06-01), Collins et al.
patent: 6417214 (2002-07-01), Ullrich et al.
patent: 6436929 (2002-08-01), Zhang et al.
patent: 6509334 (2003-01-01), Zhang et al.
patent: 6518306 (2003-02-01), Christensen
patent: 6716871 (2004-04-01), Martins et al.
patent: 2004/0002535 (2004-01-01), Fensome et al.
patent: 2004/0006060 (2004-01-01), Fensome et al.
patent: 2004/0006122 (2004-01-01), Fensome et al.
patent: 2004/0014798 (2004-01-01), Fensome et al.
patent: 314206 (1993-10-01), None
patent: WO 98/44964 (1998-10-01), None
patent: WO 00/66581 (2000-11-01), None
patent: WO 2004/000225 (2003-12-01), None
patent: WO 2004/000227 (2003-12-01), None
patent: WO 2004/000230 (2003-12-01), None
patent: WO 2004/000801 (2003-12-01), None
Fensome et al, Novel 5-Aryl-1,3-Dihydro-Indole-2-Thiones: Potent, Orally Active Progesterone Receptor Agonists, Bioorganic & Medicinal Chemistry Letters 13, pp. 1317-1320, (2003).
Testa et al, Prodrugs Revisited: The “Ad Hoc” approach as a complement to Ligand Design, Medicinal Research Reviews, 16(3):233-241, ed. John Wiley & Sons (1996).
Habte Kahsay T.
Howson & Howson LLP
Milowsky Arnold S.
Wyeth
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