Thienotriazolodiazepine compound and medicinal use thereof

Details Thienotriazolodiazepine compound and medicinal use thereof Thienotriazolodiazepine compound and medicinal use thereof

2006-05-30

2011-10-25

Coleman, Brenda (Department: 1624)

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Heterocyclic carbon compounds containing a hetero ring...

C514S220000, C540S555000, C540S560000

Reexamination Certificate

active

08044042

ABSTRACT:
A thienotriazolodiazepine compound of the following formula (I)a pharmaceutical agent containing the compound as an active ingredient, and a production intermediate and a production method of the thienotriazolodiazepine compound.Since this compound has an inhibitory action on costimulatory signal from CD28 on T cell, it is useful for the prophylaxis or suppression of rejection reaction in transplantation of organ or bone marrow and the like, and the prophylaxis or treatment of autoimmune diseases or allergic diseases.

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