Thienopyridyl compounds that inhibit vanilloid receptor...

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

Reexamination Certificate

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C546S114000

Reexamination Certificate

active

07875627

ABSTRACT:
The present invention discloses fused thienopyridyl compounds of general formula (I)wherein X1-X6, R5-R7, Z1and L are as defined in the description. The resent invention also discloses a method for inhibiting the VR1 receptor in mammals using these compounds, a method for controlling pain, urinary incontinence, bladder overactivity, and inflammatory thermal hyperalgesia in mammals, and pharmaceutical compositions including those compounds.

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