Thienodiazepines

Details Thienodiazepines Thienodiazepines

1974-03-20

1977-03-01

Thomas, Jr., James O.

Chemistry of carbon compounds

Miscellaneous organic carbon compounds

C-metal

2602948D, 2603322A, 2603323P, 2603325, 424795, C07D33324

Patent

active

040101843

ABSTRACT:
Thienodiazepines of the formula: ##STR1## wherein Ar is mono- or di-substituted phenyl [the substituents(s) being H, halogen, C.sub.1.sub.-4 alkyl or C.sub.1.sub.-4 alkoxy] or pyridyl; R.sup.1 is H or C.sub.1.sub.-4 alkyl; R.sup.2 is H, halogen or C.sub.1.sub.-4 alkyl; or R.sup.1 and R.sup.2 combinedly form -(CH.sub.2).sub.4 -; each of R.sup.3 and R.sup.4 is C.sub.1.sub.-4 alkyl, or R.sup.3 and R.sup.4 together with the adjacent nitrogen atom form a heterocyclic group; A is C.sub.2.sub.-4 alkylene; and n is an integer of zero and 1; and pharmaceutically acceptable acid addition salts thereof are disclosed. They are useful as analgesics.

REFERENCES:
masuda "Chemical Abstracts" vol. 76 (1972) p. 46225z.
Nakanishi "Journal of Medicinal Chemistry" (1973) vol. 16, No. 3, pp. 214-219.

Affiliated with

Also associated with

Rating

Thienodiazepines does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Thienodiazepines, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Thienodiazepines will most certainly appreciate the feedback.

Rate now

Comments { 0 }

Profile ID: LFUS-PAI-O-1352312