Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Reexamination Certificate
2006-10-17
2006-10-17
McKane, Joseph K. (Department: 1626)
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
C548S138000, C548S143000
Reexamination Certificate
active
07122565
ABSTRACT:
The invention provides 1,3,4-thiadiazoles and 1,3,4-oxadiazoles having the following Formula I:in which,Y is S or O,R1is alkyl, alkenyl, alkynyl, cycloalkyl, heterocycloalkyl, cycloalkenyl, aryl, heteroaryl or a polycyclic group, optionally substituted,R2is alkyl, alkenyl, alkynyl, cycloalkyl, heterocycloalkyl, cycloalkenyl or aryl optionally substituted,R3is X2—R′3, in which X2is a binding group and R′3is cycloalkyl, heterocycloalkyl, cycloalkenyl, aryl, heteroaryl, or a polycyclic group; optionally substituted, or their pharmaceutically acceptable derivatives, a compound of Formula I, for their preparation, and processes for pharmaceutical compositions containing methods of using the compounds for the treatment of disorders for which a treatment by a PDE7 inhibitor is relevant.
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Andrianjara Charles
Bernardelli Patrick
Ducrot Pierre
Ois Edwige Lorth
Vergne Fabrice
Anderson Rebecca
Benson Gregg C.
McKane Joseph K.
Richardson Peter C.
Ronau Robert T.
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