Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Patent
1995-05-19
1997-05-13
Rotman, Alan L.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
514279, 514280, 514292, 546 18, 546 41, 546 49, 546 53, 546 85, 546 86, 546 87, 546 70, A61K 3144, C07D47110, C07D48704, C07D48710
Patent
active
056293178
ABSTRACT:
The present invention provides novel tetrahydro-beta-carboline compounds having useful central nervous system activity. Further, there is provided tetrahydro-beta-carboline related compounds which are useful intermediates and have beneficial central nervous system activity. The invention provides formulations and methods for using the novel tetrahydro-beta-carboline and related compounds. Such compounds are particularly useful for the modulation of a 5-HT.sub.2B receptor.
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Audia James E.
Baker Stephen R.
Carrera Jesus E.
Peteira Carlos L.
Tercero Concepcion P.
Boone David E.
Eli Lilly and Company
Rotman Alan L.
Vorndran-Jones MaCharri R.
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