Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Patent
1997-04-09
1999-01-19
Rotman, Alan L.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
514292, 546 70, 546 86, 546 87, A61K 3144, C07D47104, C07D48704
Patent
active
058614109
ABSTRACT:
The present invention provides novel tetrahydro-beta-carboline compounds having useful central nervous system activity. Further, there is provided tetrahydro-beta-carboline related compounds which are useful intermediates and have beneficial central nervous system activity. The invention provides formulations and methods for using the novel tetrahydro-beta-carboline and related compounds. Such compounds are particularly useful for the modulation of a 5-HT.sub.2B receptor.
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Derwent Abstract 84-115276/19 Oct. 29, 1982 DE-3240-514-A.
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Audia James E.
Baker Stephen Richard
Carrera Jesus Ezquerra
Pedregal Tercero Concepcion
Peteira Carlos Lamas
Eli Lilly and Company
Palmberg Arleen
Rotman Alan L.
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