Taxanes having an amino substituted side-chain and pharmaceutica

Details Taxanes having an amino substituted side-chain and pharmaceutica Taxanes having an amino substituted side-chain and pharmaceutica

1995-06-05

1998-01-20

Trinh, Ba K.

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

549511, C07D30514

Patent

active

057102872

ABSTRACT:
Taxane derivatives having an amino substituted C13 side chain.

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G. Samaranayake et al. "Modified Taxols. 5.1 Reaction of Taxol with Electrophilic Reagents and Preparation of a Rearranged Taxol Derivative with Tubulin Assembly Activity." Journal of Organic Chemistry, 56:17, pp. 5114-5119 (1991).
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International Search Report issued for PCT/US93/10813 dated Mar. 11, 1994.

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