Organic compounds -- part of the class 532-570 series – Organic compounds – Heterocyclic carbon compounds containing a hetero ring...
Reexamination Certificate
2005-12-06
2005-12-06
Solola, Taofiq (Department: 1626)
Organic compounds -- part of the class 532-570 series
Organic compounds
Heterocyclic carbon compounds containing a hetero ring...
Reexamination Certificate
active
06972335
ABSTRACT:
The present invention provides convergent processes for preparing epothilone A and B, desoxyepothilones A and B, and analogues thereof. Also provided are analogues related to epothilone A and B and intermediates useful for preparing same. The present invention further provides novel compositions based on analogues of the epothilones and methods for the treatment of cancer and cancer which has developed a multidrug-resistant phenotype.
REFERENCES:
patent: 5021430 (1991-06-01), Ksander et al.
patent: 5917084 (1999-06-01), Jiang et al.
patent: 5969145 (1999-10-01), Schinzer et al.
patent: 6043372 (2000-03-01), Schinzer et al.
patent: 6090601 (2000-07-01), Gustafsson
patent: 6096757 (2000-08-01), Bishop
patent: 6117659 (2000-09-01), Ashley
patent: 6121029 (2000-09-01), Schupp
patent: 6156905 (2000-12-01), Schinzer et al.
patent: 6204388 (2001-03-01), Danishefsky et al.
patent: 6211412 (2001-04-01), Georg
patent: 6221641 (2001-04-01), Khosla
patent: 6242469 (2001-06-01), Danishefsky et al.
patent: 6251636 (2001-06-01), Betlach
patent: 6262094 (2001-07-01), Hoefle et al.
patent: 6262107 (2001-07-01), Li
patent: 6280999 (2001-08-01), Gustafsson
patent: 6284781 (2001-09-01), Danishefsky et al.
patent: 6288237 (2001-09-01), Hoefle et al.
patent: 6291684 (2001-09-01), Borzilleri et al.
patent: 6300355 (2001-10-01), Danishefsky et al.
patent: 6302838 (2001-10-01), O'Reilly et al.
patent: 6303342 (2001-10-01), Julien
patent: 6303767 (2001-10-01), Betlach
patent: 6316630 (2001-11-01), Danishefsky et al.
patent: 6320045 (2001-11-01), Kim et al.
patent: 6350878 (2002-02-01), Altmann
patent: 6359140 (2002-03-01), Hofle
patent: 6365749 (2002-04-01), Kim
patent: 6369234 (2002-04-01), Danishefsky
patent: 6380227 (2002-04-01), Mutz
patent: 6380394 (2002-04-01), Nicolaou
patent: 6380395 (2002-04-01), Vite
patent: 6383787 (2002-05-01), Schupp
patent: 6384230 (2002-05-01), Mulzer
patent: 6387927 (2002-05-01), Altmann
patent: 6399638 (2002-06-01), Vite
patent: 6407103 (2002-06-01), Nugiel et al.
patent: 6410301 (2002-06-01), Julien
patent: 6419692 (2002-07-01), Yang et al.
patent: 6441186 (2002-08-01), Nicolaou et al.
patent: 6457303 (2002-10-01), Georg et al.
patent: 6489314 (2002-12-01), Ashley et al.
patent: 6498257 (2002-12-01), Vite et al.
patent: 6576651 (2003-06-01), Bandyopadhyay et al.
patent: 6596875 (2003-07-01), White et al.
patent: 6670384 (2003-12-01), Bandyopadhyay et al.
patent: 6683100 (2004-01-01), Van Hoogevest
patent: 6686380 (2004-02-01), Lee
patent: 6689802 (2004-02-01), DiMarco et al.
patent: 6719540 (2004-04-01), Regueiro-Ren et al.
patent: 6723854 (2004-04-01), Danishefsky et al.
patent: 6727276 (2004-04-01), Lee
patent: 6730699 (2004-05-01), Li et al.
patent: 6730803 (2004-05-01), Iwasaki et al.
patent: 6780620 (2004-08-01), Li et al.
patent: 2001/0031880 (2001-10-01), Borzilleri et al.
patent: 2001/0034452 (2001-10-01), Hoefle et al.
patent: 2001/0051356 (2001-12-01), Khosla
patent: 2002/0002162 (2002-01-01), Lee
patent: 2002/0002194 (2002-01-01), Danishefsky et al.
patent: 2002/0004229 (2002-01-01), Santi et al.
patent: 2002/0010328 (2002-01-01), Reeves et al.
patent: 2002/0028839 (2002-03-01), O'Reilly et al.
patent: 2002/0042109 (2002-04-01), Vite et al.
patent: 2002/0045220 (2002-04-01), Khosla et al.
patent: 2002/0045609 (2002-04-01), Ashley et al.
patent: 2002/0052028 (2002-05-01), Santi et al.
patent: 2002/0058286 (2002-05-01), Danishefsky et al.
patent: 2002/0058817 (2002-05-01), Danishefsky et al.
patent: 2002/0062030 (2002-05-01), White et al.
patent: 2002/0065295 (2002-05-01), Chu et al.
patent: 2002/0086812 (2002-07-01), Schweinfest et al.
patent: 2002/0091269 (2002-07-01), Avery
patent: 2002/0115686 (2002-08-01), Hoogevest
patent: 2002/0119202 (2002-08-01), Hunter et al.
patent: 2002/0137152 (2002-09-01), Santi et al.
patent: 2002/0143038 (2002-10-01), Bandyopadhyay et al.
patent: 2002/0147197 (2002-10-01), Newman et al.
patent: 2002/0156110 (2002-10-01), Arslanian et al.
patent: 2002/0156289 (2002-10-01), Georg et al.
patent: 2002/0164377 (2002-11-01), Hunter et al.
patent: 2002/0165257 (2002-11-01), Lee
patent: 2002/0165258 (2002-11-01), Lee
patent: 2002/0165265 (2002-11-01), Hunter et al.
patent: 2002/0165415 (2002-11-01), Georg et al.
patent: 2002/0169125 (2002-11-01), Leung et al.
patent: 2002/0169135 (2002-11-01), Pardee et al.
patent: 2002/0169190 (2002-11-01), Bandyopadhyay et al.
patent: 2002/0177615 (2002-11-01), Bandyopadhyay et al.
patent: 2002/0192778 (2002-12-01), Schupp et al.
patent: 2002/0193361 (2002-12-01), Ashley et al.
patent: 2002/0197261 (2002-12-01), Li et al.
patent: 2002/0198141 (2002-12-01), McChesney et al.
patent: 2003/0003094 (2003-01-01), Hunter et al.
patent: 2003/0004209 (2003-01-01), Hunter et al.
patent: 2003/0004338 (2003-01-01), Li et al.
patent: 2003/0036177 (2003-02-01), Strohhacker
patent: 2003/0036515 (2003-02-01), Pardee et al.
patent: 2003/0045711 (2003-03-01), Ashley et al.
patent: 2003/0049841 (2003-03-01), Short et al.
patent: 2003/0054977 (2003-03-01), Kumar et al.
patent: 2003/0060623 (2003-03-01), Vite et al.
patent: 2003/0073205 (2003-04-01), Arslanian et al.
patent: 2003/0073615 (2003-04-01), Li et al.
patent: 2003/0073617 (2003-04-01), Li et al.
patent: 2003/0073677 (2003-04-01), Lee
patent: 2003/0096381 (2003-05-01), Julien et al.
patent: 2003/0105330 (2003-06-01), Danishefsky et al.
patent: 2003/0109500 (2003-06-01), Pero et al.
patent: 2003/0113335 (2003-06-01), Li et al.
patent: 2003/0114363 (2003-06-01), Li et al.
patent: 2003/0114450 (2003-06-01), Santi et al.
patent: 2003/0114504 (2003-06-01), Webster et al.
patent: 2003/0114518 (2003-06-01), Li et al.
patent: 2003/0124055 (2003-07-01), Li et al.
patent: 2003/0125362 (2003-07-01), Danishefsky et al.
patent: 2003/0130170 (2003-07-01), Li et al.
patent: 2003/0130178 (2003-07-01), Li et al.
patent: 2003/0134883 (2003-07-01), Myles et al.
patent: 2003/0139460 (2003-07-01), Schwede et al.
patent: 2003/0187273 (2003-10-01), White et al.
patent: 2003/0191089 (2003-10-01), Regueiro-Ren et al.
patent: 2004/0023345 (2004-02-01), Vite et al.
patent: 2004/0024032 (2004-02-01), Voi et al.
patent: 2004/0024033 (2004-02-01), O'Reilly et al.
patent: 2004/0030147 (2004-02-01), White et al.
patent: 2004/0038324 (2004-02-01), Atadja et al.
patent: 2004/0039026 (2004-02-01), Nicolaou et al.
patent: 2004/0044203 (2004-03-01), Wittman et al.
patent: 2004/0044221 (2004-03-01), Danishefsky et al.
patent: 2004/0049051 (2004-03-01), Hoefle et al.
patent: 2004/0053910 (2004-03-01), Danishefsky et al.
patent: 2004/0053978 (2004-03-01), Lee et al.
patent: 2004/0053995 (2004-03-01), Danishefsky et al.
patent: 2004/0054186 (2004-03-01), Das et al.
patent: 2004/0087610 (2004-05-01), Pardee et al.
patent: 2004/0087634 (2004-05-01), Hoefle et al.
patent: 2004/0092478 (2004-05-01), Rothermel et al.
patent: 2004/0092514 (2004-05-01), Velaparthi et al.
patent: 2004/0092560 (2004-05-01), Hoefle et al.
patent: 2004/0097517 (2004-05-01), Dwyer et al.
patent: 2004/0102451 (2004-05-01), Guzi et al.
patent: 2004/0102452 (2004-05-01), Guzi et al.
patent: 2004/0102495 (2004-05-01), Danishefsky et al.
patent: 2004/0106624 (2004-06-01), Guzi et al.
patent: 2004/0106985 (2004-06-01), Jang
patent: 2004/0116442 (2004-06-01), Guzi et al.
patent: 2004/0126379 (2004-07-01), Adolf et al.
patent: 2004/0127432 (2004-07-01), Nicolaou et al.
patent: 2004/0132146 (2004-07-01), Benigni et al.
patent: 2004/0132692 (2004-07-01), Sherrill et al.
patent: 2004/0132736 (2004-07-01), Guzi et al.
patent: 2004/0132754 (2004-07-01), Brandt et al.
patent: 2004/0133271 (2004-07-01), Jang
patent: 2004/0142931 (2004-07-01), Vite et al.
patent: 2004/0142990 (2004-07-01), Hofmann et al.
patent: 2004/0152708 (2004-08-01), Li et al.
patent: 41 38 042 (1991-11-01), None
patent: 19542986.9 (1995-11-01), None
patent: 196 07 702 (1996-02-01), None
patent: 196 38 870 (1996-09-01), None
patent: 19639456.2 (1996-09-01), None
patent: 197 01 758 (1997-01-01), None
patent: 197 13 970 (1997-04-01), None
patent: 19544986 (1997-05-01), None
patent: 197 20 312 (1997-05-01), None
patent: 197 26 627 (1997-06-01), None
patent: 197 35 574 (1997-0
Balog Aaron
Bertinato Peter
Chou Ting-Chao
Danishefsky Samuel J.
Kamenecka Ted
Baker C. Hunter
Choate Hall & Stewart LLP
Herschback Jarrell Brenda
Sloan-Kettering Institute for Cancer Research
Solola Taofiq
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