Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Reissue Patent
2007-01-04
2010-12-07
Sokola, Taofiq A (Department: 1625)
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
C548S204000, C548S510000, C549S271000
Reissue Patent
active
RE041990
ABSTRACT:
The present invention provides convergent processes for preparing epothilone A and B, desoxyepothilones A and B, and analogues thereof. Also provided are analogues related to epothilone A and B and intermediates useful for preparing same. The present invention further provides novel compositions based on analogues of the epothilones and methods for the treatment of cancer and cancer which has developed a multidrug-resistant phenotype.
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Balog Aaron
Bertinato Peter
Chou Ting-Chao
Danishefsky Samuel J.
Kamenecka Ted
Buteau Kristen C.
Choate Hall & Stewart LLP
Herschbach Jarrell Brenda
Sloan-Kettering Institute for Cancer Research
Sokola Taofiq A
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