Synthesis of arphamenine A

Details Synthesis of arphamenine A Synthesis of arphamenine A

1987-07-30

1989-09-26

Brust, Joseph Paul

Organic compounds -- part of the class 532-570 series

Organic compounds

Carboxylic acids and salts thereof

549415, 560 25, C07C12912

Patent

active

048702072

ABSTRACT:
Known compound, optically active arphamenine A can now be synthesized in an optically active pure form and in a favorable yield by a new process comprising consecutive steps with starting from L-arginine, wherein racemization of intermediate reaction products can be minimized.

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patent: 4595698 (1986-06-01), Umezawa et al.
House, "Modern Synthetic Reactions", 2nd ed (1972), pp. 510-511, Benjamin/Cummings Pub. Co., Menlo Park, Calif.
Royals, "Advanced Org. Chem." (1954), p. 749; Constable & Co. Ltd. London.
Rodd, "Chemistry of Carbon Compounds", (1951), (Editor), vol. 1, Part A, p. 573, Elsenies Pub. Co., London, N.Y.
McOmie (Editor) "Protective Groups in Org. Chem", 1973, Plenum Press, London & N.Y., pp. 46-47.
Meyer, et al.; J. of Med. Chem., 2y (1981), pp. 964-969.
Jennings-White, et al., Tetrahedron Letters, 23 (1982), pp. 2533-2534.

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