Sulfoximine and suldodiimine matrix metalloproteinase inhibitors

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Peptide containing doai

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2609982, 514397, 514400, 514414, 514415, 514562, 514607, 514824, 514825, 514843, 514912, 530331, 5483121, 5483131, 5483137, 5483361, 548455, 548503, A61K 3805, A61K 3806, C07K 5062, C07K 5065

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active

054708346

ABSTRACT:
Novel sulfoximine and sulfodiimine matrix metalloproteinase inhibitors of the formula, ##STR1## wherein: R.sup.1 is selected from the group consisting of lower-alkyl, hydroxy lower-alkyl, amino lower-alkyl, carbamoyl lower-alkyl, lower-alkyl carbonyl, lower-alkyoxyalkyl, aralkyl and heteroaralkyl;

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