Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Radical -xh acid – or anhydride – acid halide or salt thereof...
Reexamination Certificate
2005-01-04
2005-01-04
Barts, Samuel (Department: 1621)
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Radical -xh acid, or anhydride, acid halide or salt thereof...
C514S604000, C562S430000, C564S085000
Reexamination Certificate
active
06838483
ABSTRACT:
Compounds having a metalloproteinase inhibitory activity, represented by the formula (I), its optically active isomers, their pharmaceutically acceptable salts, or hydrates thereof.
REFERENCES:
patent: 3784701 (1974-01-01), Tomcufcik et al.
patent: 4269775 (1981-05-01), Szczepanski et al.
patent: 4388464 (1983-06-01), Kristinsson et al.
patent: 4599361 (1986-07-01), Dickens et al.
patent: 4632931 (1986-12-01), Nakane
patent: 4715883 (1987-12-01), Lukaszczyk et al.
patent: 5270326 (1993-12-01), Galardy et al.
patent: 5854277 (1998-12-01), Kluender et al.
patent: 6150394 (2000-11-01), Watanabe et al.
patent: 6207698 (2001-03-01), Wantanabe et al.
patent: 6235768 (2001-05-01), Wantanabe et al.
patent: 6441021 (2002-08-01), Wantanabe et al.
patent: 0 305 947 (1989-03-01), None
patent: 0 468 231 (1992-01-01), None
patent: 0 548 798 (1993-06-01), None
patent: 0 606 046 (1994-07-01), None
patent: 57-59969 (1982-04-01), None
patent: WO 14069 (1993-07-01), None
patent: WO 9412181 (1994-06-01), None
patent: WO 9513289 (1995-05-01), None
patent: WO 35276 (1995-12-01), None
patent: WO 9535275 (1995-12-01), None
patent: WO 9535276 (1995-12-01), None
patent: WO 00214 (1996-01-01), None
patent: WO 9600214 (1996-01-01), None
patent: WO 9611209 (1996-04-01), None
patent: WO 9615096 (1996-05-01), None
patent: WO 9727174 (1997-07-01), None
Qi-Zhuang Ye et al., Purification and Characterization of the Human Stromelysin Catalytic Domain Expressed inEscherichia coli, Biochemistry, Sep. 3, 1992, pp. 11231-11235, vol. 31-Issue No. 45, American Chemical Society.
Kevin T. Chapman et al., Inhibition of Matrix Metalloproteinases by N-Carboxyalkyl Peptides, Journal of Medicinal Chemistry, Apr. 26, 1993, pp. 4293-4301, vol. 36-Issue No. 26, American Chemical Society.
Debnath A.K., et al., “4-(4-Substituted benzoyl) aminobenzenesulphonyl-L(-)glutamic acids and 5-N-Substituted -2-[4′-(4″-substituted benzyol)aminobenzenesulphonyl]-L-glutamines as potential antineoplastic agents; Synthesis, biological evaluation and quantitative structure-activity relationsip studies,” Indian J. of Chem., 1989, pp 843-847, vol. 288.
Galli, B., et al., “Enantiomeric separation of dansyl-and dabsylamino acids by ligand-exchange chromatography with (S)- and (R)-phenylalaninamide-modified silica gel,” J. of Chroma., 1994, pp. 77-89, A.666.
Hansel J., et al., “Oxazoline Formation via a Palladium-catalyzed Cyclization: A direct, Stereoselective tocis-5-amino-2-cyclopenten-1-ol Derivatives,” 1995, Tetrahedron Letters, pp. 2913-2916, vol. 36, No. 17.
Hlavacek, J., et al, “an alternative Route to Na-Methylamino Acid Derivatives: Synthesis and Conformation of Some Na-Acetyl- Na-Methylamino Acid Methylamides,” 1988, Collect. Czechoslovak Chem. Commun., vol. 53.
Kaiser, C., et al., “2-Substituted Derivatives of 3,4-Dihydroxyphenylalanine,” 1957, pp. 4365-4370, vol. 79.
Lin, J., et al., “Debsyl Chloride: Its Synthesis, Characterization and Application in Amino Acid and Amine Microanalysis,” J. of the Chinese Biochem. Soc., 1985, pp. 10-19, vol. 14, no. 1.
Natelson, S., et al., “Preparation of D-, DL-, and L- Homoserine Lactone from Methionine,”. Microchem. Journ., 1989, pp. 226-232, vol. 40.
Nickel, P., et al., “Carboxylic acid analogues of suramin, potential filaricides,” Indian Journal of Chemistry, 1991, pp. 182-187, vol. 30B.
Stocchi, V., et al., “Reversed-Phase High Performance Liquid Chromatography Separation of Dimethylaminoazobenzene Sulfonyl-and Dimethylaminoazobenzene Thiohydantoin-Amino Acid Derivatives for Amino Acid Analysis and Microsequencing Studies at the Picomole Level,” Analyt. Biochem., 1989, pp. 107-117, vol. 178.
Verderame, M., et al., “Sulfide Derivatives of Cysteine II,” Journal of Pharma. Sci., 1962, pp 576-579, vol. 51.
Yoneda, N., et al., “Reactions of L-α-Tosylamido-β-propiolactone. I. Synthesis, Reactions with Amines and Derivation to L-Serine,” UDC, 1969, pp. 98-103, vol. 89, no. 1.
Ohtani Mitsuaki
Tsuzuki Hiroshige
Wantanabe Fumihiko
Barts Samuel
Shionogi & Co. Ltd.
LandOfFree
Sulfonated amino acid derivatives and metalloproteinase... does not yet have a rating. At this time, there are no reviews or comments for this patent.
If you have personal experience with Sulfonated amino acid derivatives and metalloproteinase..., we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Sulfonated amino acid derivatives and metalloproteinase... will most certainly appreciate the feedback.
Profile ID: LFUS-PAI-O-3372998