Drug – bio-affecting and body treating compositions – Antigen – epitope – or other immunospecific immunoeffector – Bacterium or component thereof or substance produced by said...
Patent
1983-01-21
1984-09-18
Roberts, Elbert L.
Drug, bio-affecting and body treating compositions
Antigen, epitope, or other immunospecific immunoeffector
Bacterium or component thereof or substance produced by said...
26039745, A61K 3156
Patent
active
044723920
ABSTRACT:
Novel solution stable ester prodrugs of corticosteroids of the formula ##STR1## and their salts.
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Anderson, B. D. and Taphouse, V., J. Pharm. Sci. 70 (2), Feb. 1981, pp. 181-186, "Initial Rate Studies of Hydrolysis and Acyl Migration in Methylprednisolone 21-Hemisuccinate and 17-Hemisuccinate".
Flynn, G. L. and Lamb, D. J., J. Pharm. Sci. 59 (10), Oct. 1970, pp. 1433-1438, "Factors Influencing Solvolysis of Corticosteroid-21-phosphate Esters".
Garrett, E. R., J. Pharm. Sci. 51 (5), May 1962, pp. 445-450, "Prediction of Stability in Pharmaceutical Preparations X: Alkaline Hydrolysis of Hydrocortisone Hemisuccinate".
Kawamura, M., et al., Yakugaku Zasshi, 91 (8), 1971, pp. 863-870, "Pharmaceutical Studies on Water-soluble Corticosteroid Derivatives, II. Stability of Hydrocortisone 21-Aminoalkylcarboxylates in Solution".
Kawamura, M., et al., Yakugaku Zasshi, 91 (8), 1971, pp. 871-878, "Pharmaceutical Studies on Water-soluble Corticosteroid Derivatives, III. Stability of Hydrocortisone 21-Sulfobenzoates and 21-Sulfate in Solution".
Yamamoto, R., et al., Yakugaku Zasshi, 91 (8), 1971, pp. 855-862, "Pharmaceutical Studies on Water-soluble Corticosteroid Derivatives, I. Stability of Hydrocortisone 21-Hemiesters in Solution".
Anderson Bradley D.
Conradi Robert A.
Hattan L. Ruth
Roberts Elbert L.
The Upjohn Company
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