Sulfonamides

Details Sulfonamides Sulfonamides

2011-04-26

2011-04-26

Andres, Janet L (Department: 1625)

Organic compounds -- part of the class 532-570 series

Organic compounds

Carboxylic acids and salts thereof

C562S444000, C562S506000, C514S646000, C514S659000

Reexamination Certificate

active

07932420

ABSTRACT:
The present invention provideswherein R1is selected from the group consisting of C1-C10alkoxy, OH and NR4R5;R2is selected from the group consisting of C1-C10alkyl and (CH2)nOH;R3is selected from the group consisting of C1-C10alkyl, heteroaryl, e.g. thienyl, furanyl and pyridyl, phenyl, mono, -di-, tri-substituted phenyl and heteroaryl;R4and R5are independently selected from the group consisting of H, C1-C10alkyl, C1-C10alkyl hydroxyl;m is 0 or an integer from 1 to 3 andn is an integer of from 1 to 4.These compounds are useful in lowering intraocular pressure and/or treating glaucoma or providing neuroprotection to the eye of a human patient.

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