Sulfoalkyl ether cyclodextrin based solid pharmaceutical formula

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Carbohydrate doai

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514778, 514964, 514965, 536103, A61K 31735, C07H 1312, C08B 3716

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active

058744185

ABSTRACT:
Sulfoalkyl ether-cyclodextrin (SAE-CD) based pharmaceutical formulations are provided by the present invention. These formulations comprise SAE-CD derivatives and a therapeutic agent, a major portion of which is not complexed to the SAE-CD. The present formulations are advantageously easier to prepare than other SAE-CD based formulations in the art yet provide similar or improved effectiveness. The SAE-CD derivative can be used to modify the bioavailability and/or rate of bioabsorption of therapeutic agents.

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