Substituted tyrosyl diamide compounds

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – N-c doai

Patent

Rate now

  [ 0.00 ] – not rated yet Voters 0   Comments 0

Details

514539, 514592, 514595, 514616, 560 25, 560 27, 560 34, 560 39, 564 42, 564 47, 564 56, 564153, 564157, A61K 31165, A61K 31325, A61K 3117, C07C23728

Patent

active

052721752

ABSTRACT:
The present invention provides substituted tyrosyl diamide compounds of general Formula I: ##STR1## and the pharmaceutically-acceptable salts thereof, which are useful for inducing analgesia in animals, pharmaceutical compositions comprising a pharmaceutically-acceptable carrier and a compound of Formula I, and a method for inducing analgesia in an animal in need thereof comprising administering a therapeutically-effective amount of a compound of Formula I to the animal.

REFERENCES:
patent: 4599325 (1986-07-01), Hansen, Jr. et al.
patent: 4658013 (1987-04-01), Morgan
patent: 4760180 (1988-07-01), Pitzele et al.
E. Schroder et al. Peptide Syntheses, V; Synthesis of Symmetrical etc. Liebigs Ann. Chem. 646 101-118 Jan. 1961.
R. J. Vavrek et al. Minimum Structure Opioids--Dipeptide and etc. Peptides 2 303-308 Jan. 1981.
Y. Kiso et al. Synthesis and Activity of Short-Chain etc. Peptide Chemistry 65-70 Jan. 1981.
A. R. Jacobson et al Minimum-Structure Enkephalin Analogues etc. J. Med. Chem. 32 1708-1717 Jan. 1989.
A. Guglietta et al. Dimeric Dermorphin Peptides: Central etc. Meth and Find Exp Clin Pharmacol 11(11) 663-670 Jan. 1989.

LandOfFree

Say what you really think

Search LandOfFree.com for the USA inventors and patents. Rate them and share your experience with other people.

Rating

Substituted tyrosyl diamide compounds does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Substituted tyrosyl diamide compounds, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Substituted tyrosyl diamide compounds will most certainly appreciate the feedback.

Rate now

     

Profile ID: LFUS-PAI-O-309448

  Search
All data on this website is collected from public sources. Our data reflects the most accurate information available at the time of publication.