Substituted quinolines for the treatment of protozoa and...

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

Reexamination Certificate

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C514S311000, C514S314000, C514S313000, C546S153000, C546S159000, C546S171000

Reexamination Certificate

active

10466566

ABSTRACT:
The invention relates to the use of quinolines having general formula (I), wherein R1denotes H; alkyl C1-C15; alkenyl or alkynyl C2-C15; —CHO; heteroaryl; alkyl C1-C15or alkenyl or alkynyl C2-C7comprising at least one substituent selected from among O, halogen, —OH, —CHO, —COOH, aryloxycarbonyl, alkyloxycarbonyl C2-C8, alkenyloxycarbonyl C3-C9, nitrile, aryl, heteroaryl, arylsulphone, alkylsulphone C1-C7, thioalkyl or aminoalkyl C1-C7; alkenyl C2-C7bearing at least one substituent selected from among NH2, aleoxy C1-C7, phenoxy, cycloakyl C3-C6or heteroaryloxy, alkenyl or alkynyl C2-C15comprising at least one trialkylsilyl C1-C7; R2, in position 3, 6 or 8, denotes H; halogen; —OH; —CHO; —COOH; alkyl or aleoxy C1-C7; —NH2; alkenyl C2-C7; or alkynyl C2-C10; R1and R2do not both denote H. The invention is used for the preparation of a medicine to treat protozoan and retrovirus co-infections

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