Substituted quinolin-2 (1H)-ones useful as HIV reverse transcrip

Details Substituted quinolin-2 (1H)-ones useful as HIV reverse transcrip Substituted quinolin-2 (1H)-ones useful as HIV reverse transcrip

1999-06-29

2000-07-18

Huang, Evelyn Mei

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

546158, A61K 314704, A61P 3118, C07D215227

Patent

active

060908211

ABSTRACT:
This invention relates generally to quinolin-2(1H)-ones and derivatives thereof of Formula (I): ##STR1## or stereoisomeric forms, stereoisomeric mixtures, or pharmaceutically acceptable salt forms thereof, which are useful as inhibitors of HIV reverse transcriptase, pharmaceutical compositions and diagnostic kits comprising the same, methods of using the same for treating viral infection or as assay standards or reagents, and intermediates and processes for making the same.

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