Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Reexamination Certificate
2007-11-26
2009-06-16
Saeed, Kamal A (Department: 1626)
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
C514S359000, C514S385000, C119S651000
Reexamination Certificate
active
07547718
ABSTRACT:
This invention relates to a range of alpha substituted 2-benzyl substituted imidazole compounds and pharmaceutically acceptable salts and solvates thereof, to compositions comprising such compounds, processes for their synthesis and their use as parasiticides.
REFERENCES:
patent: 4678775 (1987-07-01), Nathanson
patent: 6103733 (2000-08-01), Bachmann et al.
patent: 2005/0222135 (2005-10-01), Buschmann et al.
patent: 2006/0178404 (2006-08-01), Bowles
patent: 2007/0167506 (2007-07-01), Chubb et al.
patent: 2007/0197621 (2007-08-01), Galley et al.
patent: 2008/0119536 (2008-05-01), Chubb et al.
patent: 103 04 374 (2004-08-01), None
patent: 2 681 322 (1993-03-01), None
patent: 7-243054 (1995-09-01), None
patent: 99/28300 (1999-06-01), None
patent: 01/00586 (2001-01-01), None
patent: 01/94318 (2001-12-01), None
patent: 03/092374 (2003-11-01), None
patent: 2004/103959 (2004-12-01), None
patent: 2005/007188 (2005-01-01), None
Stella, Valentino J, Expert Opinion of Therapeutic Patents, Prodrugs as therapeutics, 2004 14(3): 277-280.
Wolff et al. (Burger's Medicinal Chemistry, 5th Ed., vol. 1, pp. 975-977, 1994).
Testa, Bernard, Biochemical Pharmacology, Prodrug Research: futile or fertile? 68 (2004) 2097-2106.
Ettmayer, Peter, Medicinal Chemistry, Lessons Learned from Marketed and Investigational Prodrugs, 47(10) (2004) 2394-2404.
PCT International Search Report, PCT/IB2007/000071.
Torregrosa et al., “Isoprene-catalyzed lithiation of imidazole: synthesis of 2-(hydroxyalkyl)- and 2-(aminoalkyl) imidazoles”, Tetrahedron, 61:11148-11155, 2005.
Nardi et al., “Research Research on durene derivatives. Note I—hypertensive activity of 2-(2,3,5,6-tetramethylbenzyl) imidazoline and related compounds”, Farmaco, Ed. Sci., 34(9):789-801, 1979.
Chubb Nathan Anthony Logan
Cox Mark Roger
Dauvergne Jerome Sebastien
Ewin Richard Andrew
Lauret Christelle
Gammill Martha A.
Pfizer Limited
Saeed Kamal A
Shterengarts Samantha L
Yang Lucy X.
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