Substituted enaminones, their derivatives and uses thereof

Details Substituted enaminones, their derivatives and uses thereof Substituted enaminones, their derivatives and uses thereof

2005-05-05

2010-11-02

Davis, Brian J (Department: 1621)

Organic compounds -- part of the class 532-570 series

Organic compounds

Amino nitrogen containing

C564S086000, C560S035000, C549S439000, C548S246000, C548S264800, C514S377000, C514S383000, C514S466000, C514S603000, C514S609000

Reexamination Certificate

active

07825278

ABSTRACT:
The invention relates to substituted enaminones of Formula I and their derivatives and the discovery that these compounds modulate the effect of γ-aminobutyric acid (GABA) on the GABAAreceptor complex in a therapeutically relevant fashion and may be used to ameliorate CNS disorders amenable to modulation of the GABAAreceptor complex.

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